Iodine-mediated one-pot synthesis of indoles and 3-dimethylaminoindoles via annulation of enaminones
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Iodine-mediated oxidative annulation for one-pot synthesis of pyrazines and quinoxalines using a multipathway coupled domino strategy.
An efficient iodine-mediated oxidative annulation of aryl acetylenes-arylethenes-aromatic ketones with 1,2-diamines for the synthesis of pyrazines and regioselective synthesis of quinoxalines is presented. A multipathway coupled domino approach has been developed for the one-pot synthesis of 1,4-diazines with high functional group compatibility.
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ژورنال
عنوان ژورنال: Arkivoc
سال: 2013
ISSN: 1551-7012
DOI: 10.3998/ark.5550190.p008.138